Proteasome
PR-924
CAS:1416709-79-9
PR-924 is a selective inhibitor of tripeptide epoxyketone immunoproteasome subunit LMP-7 (IC50: 22 nM). PR-924 …
Formula:
C37H38N4O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
618.72
Ref: TM-T16568
2mg | 670.00 € | |
1ml*10 (DMSO) | 1,704.00 € |
Estimated delivery in United States, on Thursday 23 May 2024
KZR-504
CAS:1629052-78-3
KZR-504 is a selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2) (IC50s: 51 …
Formula:
C21H23N3O6
Molecular weight:
413.42
Ref: TM-T15678
1mg | 144.00 € |
Estimated delivery in United States, on Thursday 23 May 2024
Pepstatin
CAS:26305-03-3
Pepstatin (Pepsin Inhibitor S 735A) is a specific aspartic proteases inhibitor produced by actinomycetes, and …
Formula:
C34H63N5O9
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
685.89
Ref: TM-T3695
5mg | 38.00 € | |
10mg | 52.00 € | |
25mg | 95.00 € | |
50mg | 160.00 € | |
100mg | 254.00 € | |
200mg | 369.00 € | |
1ml*10 (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Arimoclomol maleate
CAS:289893-26-1
Arimoclomol maleate (BRX-220) (BRX-220) is a heat shock protein (HSP) co-inducer.
Formula:
C18H24ClN3O7
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
429.85
Ref: TM-T13554
5mg | 46.00 € | |
10mg | 78.00 € | |
25mg | 142.00 € | |
50mg | 230.00 € | |
1ml*10 (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Retagliptin Phosphate
CAS:1256756-88-3
Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.
Formula:
C19H21F6N4O7P
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
562.36
Ref: TM-T12710
1mg | 52.00 € | |
2mg | 68.00 € | |
5mg | 96.00 € | |
10mg | 155.00 € | |
25mg | 273.00 € | |
50mg | 429.00 € | |
100mg | 584.00 € | |
1ml*10 (DMSO) | 124.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
RAMB4
CAS:145888-79-5
RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.
Formula:
C19H13Cl4NO
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
413.12
Ref: TM-T12579
10mg | 82.00 € | |
50mg | 193.00 € | |
100mg | 318.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
UT-34
CAS:2168525-92-4
UT-34 is a selective and orally active antagonist of second-generation pan-androgen receptor (AR) and degrader(IC50s …
Formula:
C15H12F4N4O2
Purity:
98.1%
Color and Shape:
Solid
Molecular weight:
356.27
Ref: TM-T13273
1mg | 52.00 € | |
2mg | 80.00 € | |
5mg | 118.00 € | |
10mg | 183.00 € | |
25mg | 425.00 € | |
50mg | 621.00 € | |
100mg | 891.00 € | |
1ml*10 (DMSO) | 129.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
DBPR108
CAS:1186426-66-3
DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no …
Formula:
C16H25FN4O2
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
324.39
Ref: TM-T15079
1mg | 115.00 € | |
5mg | 276.00 € | |
10mg | 369.00 € | |
25mg | 618.00 € | |
50mg | 878.00 € | |
100mg | 1,189.00 € | |
500mg | 2,385.00 € | |
1ml*10 (DMSO) | 304.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Sitagliptin
CAS:486460-32-6
Sitagliptin (MK0431), a new oral hypoglycemic (anti-diabetic drug), is a new dipeptidyl peptidase-4 (DPP-4) inhibitor. …
Formula:
C16H15F6N5O
Purity:
99.4%
Color and Shape:
Yellow Grease
Molecular weight:
407.31
Ref: TM-T0242
50mg | 42.00 € | |
100mg | 54.00 € | |
200mg | 64.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Aprotinin
CAS:9087-70-1
Aprotinin (Traskolan) a broad-spectrum serine protease inhibitor, inhibiting the activity of a number of different …
Formula:
C284H432N84O79S7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
6511.51
Ref: TM-T3359
5mg | 46.00 € | |
10mg | 58.00 € | |
25mg | 113.00 € | |
50mg | 184.00 € | |
100mg | 305.00 € | |
200mg | 458.00 € | |
500mg | 733.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Saxagliptin hydrate
CAS:945667-22-1
Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: …
Formula:
C18H25N3O2·H2O
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
333.43
Ref: TM-T0178
5mg | 54.00 € | |
10mg | 70.00 € | |
25mg | 117.00 € | |
50mg | 204.00 € | |
100mg | 334.00 € | |
500mg | 804.00 € | |
1ml*10 (DMSO) | 54.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Trelagliptin
CAS:865759-25-7
Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.
Formula:
C18H20FN5O2
Purity:
98.94%
Color and Shape:
Solid
Molecular weight:
357.38
Ref: TM-T6237
5mg | 53.00 € | |
10mg | 77.00 € | |
25mg | 97.00 € | |
50mg | 103.00 € | |
100mg | 135.00 € | |
1ml*10 (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Gabexate mesylate
CAS:56974-61-9
Gabexate mesylate (FOY) is a serine proteinase inhibitor used therapeutically in the treatment of pancreatitis, …
Formula:
C17H27N3O7S
Purity:
99.64%
Color and Shape:
White Crystal
Molecular weight:
417.48
Ref: TM-T0372
5mg | 55.00 € | |
10mg | 88.00 € | |
25mg | 130.00 € | |
50mg | 184.00 € | |
100mg | 301.00 € | |
200mg | 391.00 € | |
500mg | 639.00 € | |
1ml*10 (DMSO) | 73.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Racecadotril
CAS:81110-73-8
Racecadotril (Acetorphan) has been investigated for the basic science and treatment of Diarrhea, Acute Diarrhea, …
Formula:
C21H23NO4S
Purity:
99.39%
Color and Shape:
White To Off-White Crystalline Power
Molecular weight:
385.48
Ref: TM-T1176
1g | 92.00 € | |
100mg | 52.00 € | |
200mg | 57.00 € | |
500mg | 83.00 € | |
1ml*10 (DMSO) | 54.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
ML604440
CAS:1140517-08-3
ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.
Formula:
C17H24BF3N2O4
Purity:
95.24%
Color and Shape:
Solid
Molecular weight:
388.19
Ref: TM-T12079
1mg | 130.00 € | |
5mg | 268.00 € | |
10mg | 425.00 € | |
25mg | 702.00 € | |
50mg | 989.00 € | |
100mg | 1,328.00 € | |
1ml*10 (DMSO) | 295.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
RA190
CAS:1617495-03-0
RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.
Formula:
C28H23Cl5N2O2
Purity:
97.69%
Color and Shape:
Solid
Molecular weight:
596.76
Ref: TM-T13858
1mg | 56.00 € | |
5mg | 114.00 € | |
10mg | 166.00 € | |
25mg | 240.00 € | |
50mg | 427.00 € | |
100mg | 628.00 € | |
1ml*10 (DMSO) | 148.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Vildagliptin
CAS:274901-16-5
Vildagliptin (LAF237) is a cyanopyrrolidine-based, orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic …
Formula:
C17H25N3O2
Purity:
100%
Color and Shape:
White Crystalline Powder
Molecular weight:
303.4
Ref: TM-T1502
10mg | 46.00 € | |
25mg | 54.00 € | |
50mg | 66.00 € | |
100mg | 92.00 € | |
500mg | 113.00 € | |
1ml*10 (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Linagliptin
CAS:668270-12-0
Linagliptin (BI 1356) is a potent, orally bioavailable dihydropurinedione-based inhibitor of dipeptidyl peptidase 4 (DPP-4), …
Formula:
C25H28N8O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
472.54
Ref: TM-T0191
50mg | 45.00 € | |
100mg | 59.00 € | |
1ml*10 (DMSO) | 54.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
PR 39 (porcine) acetate
PR 39 (porcine) acetate is a noncompetitive, reversible and allosteric proteasome inhibitor. PR 39 (porcine) …
Purity:
98%
Molecular weight:
N/A
Ref: TM-TP1961L
1mg | To inquire | |
5mg | To inquire | |
10mg | To inquire | |
25mg | To inquire | |
50mg | To inquire |
Estimated delivery in United States, on Tuesday 28 May 2024
Calpastatin subdomain B
CAS:128578-18-7
Calpastatin subdomain B is a bioactive peptide that inhibits calpain activity.
Formula:
C140H227N35O44S
Purity:
98%
Molecular weight:
3136.57
Ref: TM-T80241
5mg | To inquire | |
50mg | To inquire |
Estimated delivery in United States, on Tuesday 28 May 2024