GRK

12 products on this category.

Product data	Purity	Price range	Estimated delivery
CMPD101 REF: TM-T14989CAS: 865608-11-3	99.01%	65.00 €~582.00 €	Tue 04 Jun 24
Paroxetine hydrochloride REF: TM-T1636CAS: 78246-49-8	99.91%	54.00 €~153.00 €	Tue 04 Jun 24
GRK6-IN-2 REF: TM-T61556CAS: 2677786-27-3	98.94%	To inquire	Mon 03 Jun 24
GSK270822A REF: TM-T27467CAS: 864082-23-5	98.77%	371.00 €~3,276.00 €	Mon 03 Jun 24
GRK2-IN-1 hydrochloride (2055990-90-2 free base) REF: TM-T13714L	98%	To inquire	Mon 03 Jun 24
GSK299115A REF: TM-T27471CAS: 864082-35-9	99.87%	314.00 €~2,759.00 €	Mon 03 Jun 24
GRK5-IN-2 REF: TM-T9609CAS: 1642839-27-7	98%	39.00 €~551.00 €	Tue 11 Jun 24
1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID REF: TM-T8913CAS: 260555-42-8	99.78%	54.00 €~401.00 €	Tue 11 Jun 24
CCG215022 REF: TM-T3498CAS: 1813527-81-9	99.69%	94.00 €~2,385.00 €	Tue 11 Jun 24
GSK180736A REF: TM-T3513CAS: 817194-38-0	98.44%	41.00 €~1,203.00 €	Tue 11 Jun 24
Takeda103A REF: TM-T24850CAS: 865609-72-9	98.01%	147.00 €~1,299.00 €	Tue 11 Jun 24
CCG258208 REF: TM-T13714CAS: 2055990-90-2	98%	1,469.00 €~4,021.00 €	Tue 03 Sep 24

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CMPD101

CAS:865608-11-3

CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM). Which …

Formula:

C₂₄H₂₁F₃N₆O

Purity:

99.01%

Color and Shape:

Solid

Molecular weight:

466.46

Ref: TM-T14989

1mg	65.00 €
5mg	124.00 €
10mg	193.00 €
25mg	389.00 €
50mg	582.00 €
1ml*10 (DMSO)	128.00 €

Estimated delivery in United States, on Tuesday 4 Jun 2024

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Paroxetine hydrochloride

CAS:78246-49-8

Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment …

Formula:

C₁₉H₂₁ClFNO₃

Purity:

99.91%

Color and Shape:

White Crystalline Powder

Molecular weight:

365.826

Ref: TM-T1636

25mg	54.00 €
50mg	63.00 €
100mg	89.00 €
200mg	113.00 €
500mg	153.00 €
1ml*10 (DMSO)	59.00 €

Estimated delivery in United States, on Tuesday 4 Jun 2024

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GRK6-IN-2

CAS:2677786-27-3

GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 …

Formula:

C₂₁H₂₁FN₆

Purity:

98.94%

Color and Shape:

Solid

Molecular weight:

376.43

Ref: TM-T61556

2mg	61.00 €
5mg	94.00 €
10mg	157.00 €
25mg	301.00 €
50mg	462.00 €
100mg	694.00 €

Estimated delivery in United States, on Monday 3 Jun 2024

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GSK270822A

CAS:864082-23-5

GSK270822A is a selective ROCK1 inhibitor. GSK270822A exhibits IC50 of 9nM, 1100nM, 1550nM for ROCK1, …

Formula:

C₂₄H₂₀N₄O₂

Purity:

98.77%

Color and Shape:

Solid

Molecular weight:

396.44

Ref: TM-T27467

1mg	371.00 €
5mg	900.00 €
10mg	1,198.00 €
25mg	1,822.00 €
50mg	2,432.00 €
100mg	3,276.00 €
1ml*10 (DMSO)	924.00 €

Estimated delivery in United States, on Monday 3 Jun 2024

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GRK2-IN-1 hydrochloride (2055990-90-2 free base)

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GRK2-IN-1 hydrochloride (2055990-90-2 free base)

GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 …

Formula:

C₂₄H₂₆ClFN₄O₄

Purity:

98%

Color and Shape:

Solid

Molecular weight:

488.94

Ref: TM-T13714L

1mg	To inquire
2mg	To inquire
5mg	To inquire
10mg	To inquire
25mg	To inquire
50mg	To inquire
100mg	To inquire
200mg	To inquire
500mg	To inquire
1ml*10 (DMSO)	To inquire

Estimated delivery in United States, on Monday 3 Jun 2024

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GSK299115A

CAS:864082-35-9

GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for …

Formula:

C₂₀H₁₆Cl₂N₄O₂

Purity:

99.87%

Color and Shape:

Solid

Molecular weight:

415.27

Ref: TM-T27471

1mg	314.00 €
5mg	755.00 €
10mg	1,054.00 €
25mg	1,560.00 €
50mg	2,107.00 €
100mg	2,759.00 €
1ml*10 (DMSO)	924.00 €

Estimated delivery in United States, on Monday 3 Jun 2024

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GRK5-IN-2

CAS:1642839-27-7

GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor. It …

Formula:

C₂₀H₂₀N₄O₄

Purity:

98%

Color and Shape:

Solid

Molecular weight:

380.4

Ref: TM-T9609

1mg	39.00 €
5mg	82.00 €
10mg	118.00 €
25mg	231.00 €
50mg	371.00 €
100mg	551.00 €
1ml*10 (DMSO)	90.00 €

Estimated delivery in United States, on Tuesday 11 Jun 2024

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1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID

CAS:260555-42-8

1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.

Formula:

C₁₃H₁₃NO₅

Purity:

99.78%

Color and Shape:

Solid

Molecular weight:

263.25

Ref: TM-T8913

5mg	54.00 €
10mg	81.00 €
25mg	123.00 €
50mg	180.00 €
100mg	267.00 €
200mg	401.00 €
1ml*10 (DMSO)	68.00 €

Estimated delivery in United States, on Tuesday 11 Jun 2024

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CCG215022

CAS:1813527-81-9

CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 …

Formula:

C₂₆H₂₂FN₇O₃

Purity:

99.69%

Color and Shape:

Solid

Molecular weight:

499.5

Ref: TM-T3498

1mg	94.00 €
2mg	138.00 €
5mg	231.00 €
10mg	369.00 €
25mg	616.00 €
50mg	877.00 €
100mg	1,196.00 €
500mg	2,385.00 €
1ml*10 (DMSO)	253.00 €

Estimated delivery in United States, on Tuesday 11 Jun 2024

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GSK180736A

CAS:817194-38-0

GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 μM) and >100-fold selectivity over …

Formula:

C₁₉H₁₆FN₅O₂

Purity:

98.44%

Color and Shape:

Solid

Molecular weight:

365.36

Ref: TM-T3513

1mg	41.00 €
2mg	52.00 €
5mg	73.00 €
10mg	87.00 €
25mg	167.00 €
50mg	300.00 €
100mg	555.00 €
500mg	1,203.00 €
1ml*10 (DMSO)	64.00 €

Estimated delivery in United States, on Tuesday 11 Jun 2024

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Takeda103A

CAS:865609-72-9

Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor.

Formula:

C₂₄H₂₃F₂N₇O

Purity:

98.01%

Color and Shape:

Solid

Molecular weight:

463.48

Ref: TM-T24850

1mg	147.00 €
5mg	276.00 €
10mg	421.00 €
25mg	690.00 €
50mg	975.00 €
100mg	1,299.00 €
1ml*10 (DMSO)	360.00 €

Estimated delivery in United States, on Tuesday 11 Jun 2024

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CCG258208

CAS:2055990-90-2

GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: …

Formula:

C₂₄H₂₅FN₄O₄

Purity:

98%

Color and Shape:

Solid

Molecular weight:

452.48

Ref: TM-T13714

25mg	2,245.00 €
50mg	2,974.00 €
100mg	4,021.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

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