Ras
In this category you can find inhibitors of Ras proteins. Ras proteins are part of the targeting process of mitogen-activated protein kinase pathways, which is a signalling pathway in eukaryotic cells.
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Opnurasib
CAS:2653994-08-0
Opnurasib (JDQ-443) is an orally available and selective and potent covalent KRAS G12C inhibitor with …
Formula:
C29H28ClN7O
Purity:
98.88%
Color and Shape:
Solid
Molecular weight:
526.03
Ref: TM-T40292
1mg | 103.00 € | |
5mg | 348.00 € | |
10mg | 517.00 € | |
25mg | 835.00 € | |
50mg | To inquire | |
1ml*10 (DMSO) | 400.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
Cysmethynil
CAS:851636-83-4
Cysmethynil is an indole-based time-dependent inhibitor of Icmt with antitumour activity and inhibitory effects on …
Formula:
C25H32N2O
Purity:
99%
Color and Shape:
Solid
Molecular weight:
376.53
Ref: TM-T36082
1mg | 46.00 € | |
2mg | 60.00 € | |
5mg | 87.00 € | |
10mg | 140.00 € | |
25mg | 273.00 € | |
50mg | 437.00 € | |
100mg | 702.00 € | |
500mg | 1,404.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
BI-2865
CAS:2937327-93-8
BI-2865 is a non-covalent pan-KRAS inhibitor.BI-2865 binds to KRAS WT, G12C, G12D, G12V, and G13D …
Formula:
C23H27N7O2S
Purity:
99.39%
Color and Shape:
Soild
Molecular weight:
465.57
Ref: TM-T72062
1mg | 212.00 € | |
5mg | 534.00 € | |
10mg | 651.00 € | |
25mg | 964.00 € | |
50mg | 1,273.00 € | |
100mg | 1,731.00 € | |
1ml*10 (DMSO) | 537.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
Digeranyl bisphosphonate
CAS:878143-03-4
Digeranyl bisphosphonate (DGBP) is a potent geranylgeranyl pyrophosphate (GGPP) synthase inhibitor that inhibits geranyl pyrophosphorylation …
Formula:
C21H34Na4O6P2
Purity:
98.50%
Color and Shape:
Solid
Molecular weight:
536.4
Ref: TM-T12452
1mg | 248.00 € | |
5mg | 499.00 € | |
10mg | 800.00 € | |
25mg | 1,410.00 € | |
50mg | 1,846.00 € | |
100mg | 2,322.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
BI-0474
CAS:2750570-55-7
BI-0474 is a potent KRASG12C inhibitor that inhibits GDP-KRAS::SOS1 protein-protein interactions with an IC50 value …
Formula:
C30H37N9O2S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
587.74
Ref: TM-T69529
1mg | 403.00 € | |
5mg | 920.00 € | |
10mg | 1,277.00 € | |
25mg | 1,846.00 € | |
50mg | 2,545.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
Deltarasin
CAS:1440898-61-2
Deltarasin is a small molecular inhibitor of KRAS-PDEδ interaction with Kd of 38 nM for …
Formula:
C40H37N5O
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
603.75
Ref: TM-T6462
1mg | 48.00 € | |
2mg | 64.00 € | |
5mg | 118.00 € | |
10mg | 185.00 € | |
25mg | To inquire | |
50mg | To inquire | |
1ml*10 (DMSO) | 158.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
MCP110
CAS:521310-51-0
MCP110 is an inhibitor of the interaction of Ras with Raf-1 and can be used …
Formula:
C33H36N2O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
508.65
Ref: TM-T24437
1mg | 72.00 € | |
5mg | 158.00 € | |
10mg | 267.00 € | |
25mg | 475.00 € | |
50mg | 690.00 € | |
100mg | 922.00 € | |
500mg | 1,839.00 € | |
1ml*10 (DMSO) | 171.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
BI-2852
CAS:2375482-51-0
BI-2852 is a KRAS inhibitor for the switch I/II pocket (SI/II-pocket) with nanomolar affinity. BI-2852 …
Formula:
C31H28N6O2
Purity:
98.98%
Color and Shape:
Solid
Molecular weight:
516.59
Ref: TM-T10533
1mg | 115.00 € | |
5mg | 271.00 € | |
10mg | 401.00 € | |
25mg | 664.00 € | |
50mg | 916.00 € | |
100mg | 1,263.00 € | |
1ml*10 (DMSO) | 311.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
TH-Z827
CAS:2847881-81-4
TH-Z827 is a mutant-selective inhibitor targeting KRAS(G12D) with an IC50 of 2.4 μM, demonstrating specificity …
Formula:
C30H38N6O
Purity:
98%
Molecular weight:
498.66
Ref: TM-T79092
5mg | To inquire | |
50mg | To inquire |
Estimated delivery in United States, on Monday 3 Jun 2024
Ras Inhibitory Peptide acetate
Ras Inhibitory Peptide acetate is a peptide involved in the Ras-dependent signaling pathway that plays …
Formula:
C55H95N19O13
Purity:
96.63%
Color and Shape:
Solid
Molecular weight:
1230.46
Ref: TM-T37422L
1mg | 182.00 € | |
5mg | 409.00 € | |
10mg | 600.00 € | |
25mg | 917.00 € | |
50mg | 1,281.00 € | |
100mg | 1,733.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
CCG-257081
CAS:1922098-90-5
CCG-257081 (MRTF/SRF-IN-1) is an inhibitor of cardiac myosin-related transcription factor and serum response factor (MRTF/SRF) …
Formula:
C24H19ClF3N3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
473.87
Ref: TM-T30778
1mg | 125.00 € | |
5mg | 293.00 € | |
10mg | 435.00 € | |
25mg | 714.00 € | |
50mg | 1,000.00 € | |
100mg | 1,346.00 € | |
500mg | 2,685.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
(E/Z)-ZINC09659342
CAS:591726-26-0
(E/Z)-ZINC09659342 is an inhibitor of Lbc-Rho A interaction.
Formula:
C23H15F3N2O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
440.37
Ref: TM-T9986
1mg | 121.00 € | |
5mg | 292.00 € | |
10mg | 464.00 € | |
25mg | 737.00 € | |
50mg | 1,054.00 € | |
100mg | 1,417.00 € | |
500mg | 2,757.00 € | |
1ml*10 (DMSO) | 321.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
KRAS G12C inhibitor 19
CAS:2649788-46-3
KRAS G12C inhibitor 19 is a potent KRAS G12C inhibitor that shows anti-tumor activity in …
Formula:
C25H19ClF2N4O3S
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
528.96
Ref: TM-T40286
1mg | 89.00 € | |
5mg | 182.00 € | |
10mg | 274.00 € | |
25mg | 532.00 € | |
50mg | 765.00 € | |
100mg | 1,050.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
LUNA18
CAS:2676177-63-0
LUNA18 is an orally active inhibitor targeting KRAS, exhibiting potent activity with an IC50 value …
Formula:
C73H105F5N12O12
Purity:
98%
Molecular weight:
1437.68
Ref: TM-T79673
5mg | To inquire | |
50mg | To inquire |
Estimated delivery in United States, on Monday 3 Jun 2024
KRAS G12D modulator-1
CAS:2883034-05-5
KRAS G12D modulator-1 (compound 6), a potent modulator of KRAS G12D, exhibits IC50 values ranging …
Formula:
C30H36FN5O4
Purity:
98%
Molecular weight:
549.64
Ref: TM-T79072
5mg | To inquire | |
50mg | To inquire |
Estimated delivery in United States, on Monday 3 Jun 2024
Kras4B G12D-IN-1
CAS:2042365-85-3
Kras4B G12D-IN-1 is an anticancer agent that functions as an inhibitor of the Kras4B G12D …
Formula:
C16H21ClN2O4S
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
372.87
Ref: TM-T78170
2mg | 96.00 € | |
5mg | 150.00 € | |
10mg | 238.00 € | |
25mg | 483.00 € | |
50mg | 772.00 € | |
100mg | 1,175.00 € | |
500mg | 2,359.00 € | |
1ml*10 (DMSO) | 167.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
BI-2493
CAS:2937344-16-4
BI-2493 is a highly selective pan-KRAS inhibitor and structural analog of BI-2865.BI-2493 exhibits antitumor activity …
Formula:
C24H27N7OS
Purity:
99.49%
Color and Shape:
Soild
Molecular weight:
461.58
Ref: TM-T72061
1mg | 587.00 € | |
5mg | 1,444.00 € | |
10mg | 2,300.00 € | |
25mg | 3,413.00 € | |
50mg | 4,545.00 € | |
100mg | 6,149.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
KRAS G12C inhibitor 58
CAS:2915599-52-7
KRAS G12C inhibitor 58 is utilized in cancer research as an inhibitor of the KRAS …
Formula:
C51H64ClF4N9O8S
Purity:
98%
Molecular weight:
1074.62
Ref: TM-T79057
5mg | To inquire | |
50mg | To inquire |
Estimated delivery in United States, on Monday 3 Jun 2024
SOS1-IN-11
CAS:2654741-64-5
SOS1-IN-11 is an effective inhibitor of SOS1 (IC50 = 30 nM).
Formula:
C22H24F3N5O
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
431.45
Ref: TM-T60029
1mg | 112.00 € | |
5mg | 270.00 € | |
10mg | 465.00 € | |
25mg | 740.00 € | |
50mg | 1,054.00 € | |
100mg | 1,411.00 € | |
1ml*10 (DMSO) | 295.00 € |
Estimated delivery in United States, on Monday 3 Jun 2024
Rac1-IN-3
CAS:380470-06-4
Rac1-IN-3 (Compound 2) is a Rac1 inhibitor exhibiting an inhibitory concentration 50 (IC50) of 46.1 …
Formula:
C21H23N7O2
Purity:
98%
Molecular weight:
405.45
Ref: TM-T79869
5mg | To inquire | |
50mg | To inquire |
Estimated delivery in United States, on Monday 3 Jun 2024