Ras
In this category you can find inhibitors of Ras proteins. Ras proteins are part of the targeting process of mitogen-activated protein kinase pathways, which is a signalling pathway in eukaryotic cells.
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CCG-203971
CAS:1443437-74-8
CCG-203971 is an inhibitor of SRE activation in the prostate cancer cell line PC-3 (IC50: …
Formula:
C23H21ClN2O3
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
408.88
Ref: TM-T4306
10mg | 53.00 € | |
25mg | 94.00 € | |
50mg | 144.00 € | |
100mg | 224.00 € | |
500mg | 553.00 € | |
1ml*10 (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
ML141
CAS:71203-35-5
ML141 (CID-2950007) is an effective, specific and reversible non-competitive inhibitor of Rho family GTPase cdc42 …
Formula:
C22H21N3O3S
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
407.49
Ref: TM-T2463
1mg | 39.00 € | |
2mg | 50.00 € | |
5mg | 71.00 € | |
10mg | 108.00 € | |
25mg | 219.00 € | |
50mg | 398.00 € | |
100mg | 568.00 € | |
500mg | 1,226.00 € | |
1ml*10 (DMSO) | 74.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
ARS-1620
CAS:1698055-85-4
ARS-1620 is a covalent inhibitor of K-RASG12C.
Formula:
C21H17ClF2N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
430.84
Ref: TM-T7609
1mg | 90.00 € | |
2mg | 115.00 € | |
5mg | 185.00 € | |
10mg | 269.00 € | |
25mg | 531.00 € | |
50mg | 763.00 € | |
100mg | 916.00 € | |
1ml*10 (DMSO) | 209.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
Rasarfin
CAS:674359-73-0
Rasarfin inhibits Ras and ARF6.
Formula:
C23H24ClN3O3
Purity:
98.58%
Color and Shape:
Solid
Molecular weight:
425.91
Ref: TM-T9407
1mg | 61.00 € | |
2mg | 85.00 € | |
5mg | 118.00 € | |
10mg | 184.00 € | |
25mg | 335.00 € | |
50mg | 557.00 € | |
100mg | 794.00 € | |
500mg | 1,612.00 € | |
1ml*10 (DMSO) | 129.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
Atranorin
CAS:479-20-9
Atranorin shows significant antinociceptive and antiinflammatory activities, it has a relevant redox-active action, acting as …
Formula:
C19H18O8
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
374.34
Ref: TM-TN1413
1mg | 105.00 € | |
5mg | 247.00 € | |
10mg | 365.00 € | |
25mg | 612.00 € | |
50mg | 873.00 € | |
100mg | 1,180.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
CASIN
CAS:425399-05-9
CASIN (Pirl1-related Compound 2) is a specific inhibitor of GTPase Cdc42 (IC50: 2 uM).
Formula:
C20H22N2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
306.4
Ref: TM-T3971
1mg | 38.00 € | |
2mg | 49.00 € | |
5mg | 74.00 € | |
10mg | 119.00 € | |
25mg | 184.00 € | |
50mg | 276.00 € | |
100mg | 425.00 € | |
500mg | 916.00 € | |
1ml*10 (DMSO) | 73.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
EHT 1864
CAS:754240-09-0
EHT 1864 is a effective Rac family GTPase inhibitor for Rac1/Rac1b/Rac2/Rac3 (Kd: 40/50/60/250 nM).
Formula:
C25H29Cl2F3N2O4S
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
581.47
Ref: TM-T6483
1mg | 46.00 € | |
5mg | 90.00 € | |
10mg | 134.00 € | |
25mg | 254.00 € | |
50mg | 464.00 € | |
100mg | 666.00 € | |
200mg | 917.00 € | |
1ml*10 (DMSO) | 105.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
Kobe0065
CAS:436133-68-5
Kobe0065 is a novel and effective small-molecule compound inhibiting Ras-Raf interaction by SBDD; shows potent …
Formula:
C15H11ClF3N5O4S
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
449.79
Ref: TM-T1876
5mg | 46.00 € | |
10mg | 62.00 € | |
25mg | 95.00 € | |
50mg | 139.00 € | |
100mg | 217.00 € | |
200mg | 361.00 € | |
500mg | 600.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
FTI-277 hydrochloride
CAS:180977-34-8
FTI-277 hydrochloride (FTI 277 HCl) is an effective and specific farnesyltransferase (FTase) inhibitor (IC50: 500 …
Formula:
C22H30ClN3O3S2
Purity:
98.19%
Color and Shape:
Solid
Molecular weight:
484.07
Ref: TM-T2700
1mg | 52.00 € | |
2mg | 77.00 € | |
5mg | 99.00 € | |
10mg | 177.00 € | |
25mg | 318.00 € | |
50mg | 530.00 € | |
100mg | 742.00 € | |
1ml*10 (DMSO) | 109.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
(S)-AMG-510
CAS:2252403-56-6
(S)-AMG-510 is an S-type compound of AMG-510, a potent covalent inhibitor of KRAS G12C with …
Formula:
C30H30F2N6O3
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
560.59
Ref: TM-T22258
2mg | 36.00 € | |
5mg | 52.00 € | |
10mg | 83.00 € | |
25mg | 152.00 € | |
50mg | 268.00 € | |
100mg | 420.00 € | |
500mg | 917.00 € | |
1ml*10 (DMSO) | 75.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
K-Ras(G12C) inhibitor 12
CAS:1469337-95-8
K-Ras(G12C) inhibitor 12 is an allosteric inhibitor of oncogenic K-Ras(G12C).
Formula:
C15H17ClIN3O3
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
449.67
Ref: TM-T6555
1mg | 52.00 € | |
2mg | 73.00 € | |
5mg | 113.00 € | |
10mg | 184.00 € | |
25mg | 305.00 € | |
50mg | 454.00 € | |
100mg | 666.00 € | |
1ml*10 (DMSO) | 123.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
ERK-IN-3
CAS:2055597-12-9
ERK-IN-3 (ASN007 free base) is a potent and orally active inhibitor of ERK. It inhibits …
Formula:
C22H25ClFN7O2
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
473.93
Ref: TM-T9141
1mg | 60.00 € | |
5mg | 122.00 € | |
10mg | 172.00 € | |
25mg | 280.00 € | |
50mg | 457.00 € | |
1ml*10 (DMSO) | 124.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
ASP2453
CAS:2241719-73-1
ASP2453 is a potent, selective and covalent inhibitor of KRAS G12C. ASP2453 inhibits the Son …
Formula:
C40H48F3N7O4
Purity:
96.57%
Color and Shape:
Solid
Molecular weight:
747.85
Ref: TM-T39738
1mg | 183.00 € | |
5mg | 477.00 € | |
10mg | 694.00 € | |
25mg | 1,077.00 € | |
50mg | 1,449.00 € | |
1ml*10 (DMSO) | 712.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
CCG-1423
CAS:285986-88-1
CCG-1423, a selective RhoA pathway inhibitor, suppresses SRF-mediated transcription.
Formula:
C18H13ClF6N2O3
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
454.75
Ref: TM-T2014
5mg | 38.00 € | |
10mg | 56.00 € | |
25mg | 94.00 € | |
50mg | 159.00 € | |
100mg | 256.00 € | |
200mg | 399.00 € | |
500mg | 646.00 € | |
1ml*10 (DMSO) | 54.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
6H05 (TFA)
CAS:2061344-88-3
6H05 TFA (6H05 trifluoroacetate) is a selective, and allosteric oncogenic mutant K-Ras(G12C) inhibitor.
Formula:
C22H31ClF3N3O4S3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
590.14
Ref: TM-T7326
1mg | 68.00 € | |
2mg | 94.00 € | |
5mg | 131.00 € | |
10mg | 225.00 € | |
25mg | 369.00 € | |
50mg | 559.00 € | |
100mg | 789.00 € | |
1ml*10 (DMSO) | 171.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
Compound 3344 hydrochloride
Compound 3344 hydrochloride is an inhibitor of KRAS-effector interactions,with an affnity of 126nm.
Formula:
C24H27ClN2O3
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
426.94
Ref: TM-T9184L
1mg | 141.00 € | |
5mg | 278.00 € | |
10mg | 416.00 € | |
25mg | 686.00 € | |
50mg | 920.00 € | |
100mg | 1,287.00 € | |
1ml*10 (DMSO) | 330.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
SCH54292
CAS:188480-51-5
SCH-54292 is a GDP exchange inhibitor.
Formula:
C24H28N2O9S
Purity:
95.65%
Color and Shape:
Solid
Molecular weight:
520.55
Ref: TM-T9198
1mg | 129.00 € | |
5mg | 282.00 € | |
10mg | 420.00 € | |
25mg | 692.00 € | |
50mg | 975.00 € | |
1ml*10 (DMSO) | 356.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
ZT-12-037-01
CAS:2328073-61-4
Zt-12-037-01 is a ATP competitive STK19 inhibitor(IC50 values of 23.96 nM and 27.94 nM for …
Formula:
C21H31N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
385.5
Ref: TM-T5597
1mg | 35.00 € | |
2mg | 52.00 € | |
5mg | 73.00 € | |
10mg | 113.00 € | |
25mg | 221.00 € | |
50mg | 425.00 € | |
100mg | 629.00 € | |
1ml*10 (DMSO) | 81.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
BAY-293
CAS:2244904-70-7
BAY-293 is a potent, cell-active SOS1 inhibitor that disrupts the KRAS-SOS1 interaction (IC50: 21 nM).
Formula:
C25H28N4O2S
Purity:
96.8%
Color and Shape:
Solid
Molecular weight:
448.58
Ref: TM-T5418
1mg | 52.00 € | |
5mg | 109.00 € | |
10mg | 183.00 € | |
25mg | 368.00 € | |
50mg | 547.00 € | |
100mg | 786.00 € | |
1ml*10 (DMSO) | 121.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024
(Rac)-Antineoplaston A10
CAS:77658-84-5
(Rac)-Antineoplaston A10 (Antineoplaston A10) is a naturally occurring substance and the first antineoplaston in the …
Formula:
C13H14N2O3
Purity:
98.47%
Color and Shape:
Solid
Molecular weight:
246.26
Ref: TM-T5379
1mg | 60.00 € | |
2mg | 95.00 € | |
5mg | 129.00 € | |
10mg | 204.00 € | |
25mg | 341.00 € | |
50mg | 507.00 € | |
100mg | 731.00 € | |
1ml*10 (DMSO) | 140.00 € |
Estimated delivery in United States, on Tuesday 11 Jun 2024